![]() |
GF-109203X
- 英文名称:GF-109203X
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10020
- cas:133052-90-1
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10020 |
用途 | 科研检测 |
英文名称 | GF-109203X |
包装规格 | 1MG |
CAS编号 | 133052-90-1 |
别名 | GF-109203X |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC NMR conforms
分子式:C25H24N4O2
分子量:412.49
溶剂:DMSO (10 mg/ml)
性状:Orange solid
存储:RT
Activity (short version):PKC inhibitor
Function / Pharmacology:Potent and selective protein kinase C inhibitor (IC50 = 10 nM; cAMP-dependent protein kinase IC50 = 2 μM and phosphorylase kinase IC50 = 0.7 μM). Inactive against the tyrosine kinases EGFR, PGDFR and Insulin receptor. Potent inhibitor of GSK-3β in cell lysates (IC50 = 360nM) and GSK-3β immunoprecipitates (IC50 = 170nM) derived from rat epididymal adipocytes.2 Cell permeable.
分子式:C25H24N4O2
分子量:412.49
溶剂:DMSO (10 mg/ml)
性状:Orange solid
存储:RT
Activity (short version):PKC inhibitor
Function / Pharmacology:Potent and selective protein kinase C inhibitor (IC50 = 10 nM; cAMP-dependent protein kinase IC50 = 2 μM and phosphorylase kinase IC50 = 0.7 μM). Inactive against the tyrosine kinases EGFR, PGDFR and Insulin receptor. Potent inhibitor of GSK-3β in cell lysates (IC50 = 360nM) and GSK-3β immunoprecipitates (IC50 = 170nM) derived from rat epididymal adipocytes.2 Cell permeable.