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A-803467
- 英文名称：A-803467
- 品牌：WYTSCI
- 产地：进口
- 型号：1MG
- 货号：WT-AY-B10056
- cas：944261-79-4
- 价格： ￥1/mg
- 发布日期： 2025-04-10
- 更新日期： 2025-12-08
产品详请
| 产地 | 进口 |
| 品牌 | WYTSCI |
| 货号 | WT-AY-B10056 |
| 用途 | 科研检测 |
| 英文名称 | A-803467 |
| 包装规格 | 1MG |
| CAS编号 | 944261-79-4 |
| 别名 | A-803467 |
| 纯度 | 98+% |
| 分子式 | |
| 是否进口 | 是 |
纯度:98% by TLC [50% ethyl acetate in hexanes, Rf = 0.58] NMR Conforms
分子式:C19H16ClNO4
分子量:357.80
溶剂:DMSO (15 mg/ml) Ethanol (2 mg/ml)
性状:white solid (MP = 128-130°C)
存储:RT
Activity (short version):NaV1.8 blocker
Function / Pharmacology:Potent, selective inhibitor of the TTX-resistant voltage-gated sodium channel Nav1.8. Nav1.8 is preferentially expressed in sensory neurons, and inhibition attenuates both inflammatory and neuropathic pain in a variety of animal models. IC50's for rat and human Nav1.8 are 140 nM and 8.0 nM respectively.
分子式:C19H16ClNO4
分子量:357.80
溶剂:DMSO (15 mg/ml) Ethanol (2 mg/ml)
性状:white solid (MP = 128-130°C)
存储:RT
Activity (short version):NaV1.8 blocker
Function / Pharmacology:Potent, selective inhibitor of the TTX-resistant voltage-gated sodium channel Nav1.8. Nav1.8 is preferentially expressed in sensory neurons, and inhibition attenuates both inflammatory and neuropathic pain in a variety of animal models. IC50's for rat and human Nav1.8 are 140 nM and 8.0 nM respectively.
