纯度:98% by HPLC;NMR (Conforms)
分子式:C19H35N3O4S
分子量:401.56
溶剂:DMSO (10 mg/ml) Ethanol (5 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):Calpain inhibitor
Function / Pharmacology:Cell-permeable, peptide aldehyde inhibitor of calpain (calpain I, Ki = 120 nM, calpain II, Ki = 230 nM) and other neutral cysteine proteases. Potent inhibitor of cathepsin L (Ki=0.6 nM) and cathepsin B (Ki=100 nM).1 Weak inhibitor of the chymotrypsin-like activity of the proteasome.2 Cell permeable.