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WP-1130
- 英文名称:WP-1130
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10255
- cas:856243-80-6
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-12
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10255 |
用途 | 科研检测 |
英文名称 | WP-1130 |
包装规格 | 1MG |
CAS编号 | 856243-80-6 |
别名 | WP-1130 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC,;NMR (Conforms)
分子式:C19H18BrN3O
分子量:384.28
溶剂:DMSO (45 mg/ml) Ethanol (25 mg/ml)
性状:Yellow solid
存储:-20°C
Activity (short version):DUB inhibitor
Function / Pharmacology:A novel DUB inhibitor directly inhibiting USP9x, USP5, USP14 and UCH37 inducing rapid accumulation of polyubiquitinated proteins. Triggers tumor cell apoptosis.1 Blocks Jak2 signaling via Jak2 ubiquitination.2 Causes ablation of the oncogenic transcription factor ERG in prostate cancer cells.3
分子式:C19H18BrN3O
分子量:384.28
溶剂:DMSO (45 mg/ml) Ethanol (25 mg/ml)
性状:Yellow solid
存储:-20°C
Activity (short version):DUB inhibitor
Function / Pharmacology:A novel DUB inhibitor directly inhibiting USP9x, USP5, USP14 and UCH37 inducing rapid accumulation of polyubiquitinated proteins. Triggers tumor cell apoptosis.1 Blocks Jak2 signaling via Jak2 ubiquitination.2 Causes ablation of the oncogenic transcription factor ERG in prostate cancer cells.3