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MRL-24
- 英文名称:MRL-24
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10267
- cas:393794-17-7
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10267 |
用途 | 科研检测 |
英文名称 | MRL-24 |
包装规格 | 1MG |
CAS编号 | 393794-17-7 |
别名 | MRL-24 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC,;NMR (Conforms)
分子式:C28H24F3NO6
分子量:527.49
溶剂:DMSO (30 mg/ml)
性状:White solid
存储:RT
Activity (short version):PPARγ partial agonist
Function / Pharmacology:Displays high affinity for PPARγ with excellent anti-diabetic activity in mice but poor PPARγ agonist activity in transcription and adipogenesis assays. Highly effective (30 nM) at blocking Cdk5-mediated phosphorylation of PPARγ. Cell permeable.
分子式:C28H24F3NO6
分子量:527.49
溶剂:DMSO (30 mg/ml)
性状:White solid
存储:RT
Activity (short version):PPARγ partial agonist
Function / Pharmacology:Displays high affinity for PPARγ with excellent anti-diabetic activity in mice but poor PPARγ agonist activity in transcription and adipogenesis assays. Highly effective (30 nM) at blocking Cdk5-mediated phosphorylation of PPARγ. Cell permeable.