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TC-E 5003
- 英文名称:TC-E 5003
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10374
- cas:17328-16-4
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-16
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10374 |
用途 | 科研检测 |
英文名称 | TC-E 5003 |
包装规格 | 1MG |
CAS编号 | 17328-16-4 |
别名 | TC-E 5003 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by HPLC;NMR (Conforms)
分子式:C16H14Cl2N2O4S
分子量:401.26
溶剂:DMSO 50 mg/ml
性状:Brown solid
存储:-20°C
Activity (short version):Arginine methyl transferase 1 (PRMT1) inhibitor
Function / Pharmacology:Selective protein arginine methyltransferase 1 (PRMT1) inhibitor, IC50 = 1.5 μM. Displays no activity against CARM1 and Set7/9 methyltransferases. Inhibits growth of MCF7a breast cancer cells and LNCaP prostate cancer cells. Blocks androgen-induced gene expression in LNCaP cells1.
分子式:C16H14Cl2N2O4S
分子量:401.26
溶剂:DMSO 50 mg/ml
性状:Brown solid
存储:-20°C
Activity (short version):Arginine methyl transferase 1 (PRMT1) inhibitor
Function / Pharmacology:Selective protein arginine methyltransferase 1 (PRMT1) inhibitor, IC50 = 1.5 μM. Displays no activity against CARM1 and Set7/9 methyltransferases. Inhibits growth of MCF7a breast cancer cells and LNCaP prostate cancer cells. Blocks androgen-induced gene expression in LNCaP cells1.