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YM-254890
- 英文名称:YM-254890
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10435
- cas:568580-02-9
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-12
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10435 |
用途 | 科研检测 |
英文名称 | YM-254890 |
包装规格 | 1MG |
CAS编号 | 568580-02-9 |
别名 | YM-254890 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:95% by HPLC,;NMR (Conforms)
分子式:C46H69N7O15
分子量:960.10
溶剂:DMSO (10 mg/ml)
性状:White or off-white lyophilize solid
存储:-20°C
Activity (short version):Gq inhibitor
Function / Pharmacology:YM-254890 is a novel Gαq/11 inhibitor,1 U46619-induced platelet aggregation is inhibited but phorbol ester- or ionophore-induced aggregation is not2 (IC50 = 0.1-0.2 μM)1. It blocks Pasteurella multocida toxin-mediated activation of Gαq.3 A highly useful new tool for studying Gαq/11-coupled receptor signaling and resulting cellular events.4
分子式:C46H69N7O15
分子量:960.10
溶剂:DMSO (10 mg/ml)
性状:White or off-white lyophilize solid
存储:-20°C
Activity (short version):Gq inhibitor
Function / Pharmacology:YM-254890 is a novel Gαq/11 inhibitor,1 U46619-induced platelet aggregation is inhibited but phorbol ester- or ionophore-induced aggregation is not2 (IC50 = 0.1-0.2 μM)1. It blocks Pasteurella multocida toxin-mediated activation of Gαq.3 A highly useful new tool for studying Gαq/11-coupled receptor signaling and resulting cellular events.4