![]() |
Erlotinib · HCl
- 英文名称:Erlotinib · HCl
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10546
- cas:183319-69-9
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10546 |
用途 | 科研检测 |
英文名称 | Erlotinib · HCl |
包装规格 | 1MG |
CAS编号 | 183319-69-9 |
别名 | Erlotinib · HCl |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC,;NMR (Conforms)
分子式:C22H23N3O4 · HCl
分子量:429.91
溶剂:DMSO (18 mg/ml)
性状:White or off-white solid
存储:-20°C
Activity (short version):EGFR Kinase inhibitor
Function / Pharmacology:Potent inhibitor of EGFR tyrosine kinase (IC50 = 2 nM)1. Potent inhibitor of mutant JAK2-V617F2. Weaker inhibitor of ErbB-2 kinase (Ki = 1 μM) ErbB-4 kinase (Ki = 1.5 μM)3. HDAC inhibitors sensitize for erlotinib activity in EGFR-mutated and wildtype non-small cell lung cancer (NSCLC) cells4. A clinically effective agent for NSCLC5.
分子式:C22H23N3O4 · HCl
分子量:429.91
溶剂:DMSO (18 mg/ml)
性状:White or off-white solid
存储:-20°C
Activity (short version):EGFR Kinase inhibitor
Function / Pharmacology:Potent inhibitor of EGFR tyrosine kinase (IC50 = 2 nM)1. Potent inhibitor of mutant JAK2-V617F2. Weaker inhibitor of ErbB-2 kinase (Ki = 1 μM) ErbB-4 kinase (Ki = 1.5 μM)3. HDAC inhibitors sensitize for erlotinib activity in EGFR-mutated and wildtype non-small cell lung cancer (NSCLC) cells4. A clinically effective agent for NSCLC5.