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Obatoclax
- 英文名称:Obatoclax
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10760
- cas:803712-79-0
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10760 |
用途 | 科研检测 |
英文名称 | Obatoclax |
包装规格 | 1MG |
CAS编号 | 803712-79-0 |
别名 | Obatoclax |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC
分子式:C20H19N3O · CH3SO3H
分子量:413.50
溶剂:DMSO (5 mg/ml)
性状:Purple solid
存储:-20°C
Activity (short version):BCL-2 antagonist; Induces apoptosis
Function / Pharmacology:A novel Bcl-2 homology domain-3 (BH3) mimetic1. Inhibits primary acute myeloid leukemia (AML) progenitor cell proliferation (IC50=0.18 μM) and induces apoptosis in primary AML cells (IC50= 3.6 μM)2. Synergizes with other agents such as chloroquine3 and cytarabine4 in cytotoxicity against a variety of cancer cells.
分子式:C20H19N3O · CH3SO3H
分子量:413.50
溶剂:DMSO (5 mg/ml)
性状:Purple solid
存储:-20°C
Activity (short version):BCL-2 antagonist; Induces apoptosis
Function / Pharmacology:A novel Bcl-2 homology domain-3 (BH3) mimetic1. Inhibits primary acute myeloid leukemia (AML) progenitor cell proliferation (IC50=0.18 μM) and induces apoptosis in primary AML cells (IC50= 3.6 μM)2. Synergizes with other agents such as chloroquine3 and cytarabine4 in cytotoxicity against a variety of cancer cells.