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ML204
- 英文名称:ML204
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B10826
- cas:5465-86-1
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B10826 |
用途 | 科研检测 |
英文名称 | ML204 |
包装规格 | 1MG |
CAS编号 | 5465-86-1 |
别名 | ML204 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC,;NMR (Conforms)
分子式:C15H18N2
分子量:226.32
溶剂:DMSO (20 mg/ml)
性状:Off-white solid
存储:-20°C
Activity (short version):TRPC4 blocker
Function / Pharmacology:Selective blocker of TRPC4 channels (IC50 = 0.96 - 2.6 μM, depending on assay). Displays 19-fold selectivity against TRPC6 and 9-fold selectivity against TRPC5. Has no significant activity at TRPV1, TRPV3, TRPA1 and TRPM8 channels at concentrations up to 22 μM. A useful tool for exploring the involvement of TRPC and TRPC-like channels in cellular signaling and physiology.2-4
分子式:C15H18N2
分子量:226.32
溶剂:DMSO (20 mg/ml)
性状:Off-white solid
存储:-20°C
Activity (short version):TRPC4 blocker
Function / Pharmacology:Selective blocker of TRPC4 channels (IC50 = 0.96 - 2.6 μM, depending on assay). Displays 19-fold selectivity against TRPC6 and 9-fold selectivity against TRPC5. Has no significant activity at TRPV1, TRPV3, TRPA1 and TRPM8 channels at concentrations up to 22 μM. A useful tool for exploring the involvement of TRPC and TRPC-like channels in cellular signaling and physiology.2-4