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BAY-1797
- 英文名称:BAY-1797
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11042
- cas:2055602-83-8
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11042 |
用途 | 科研检测 |
英文名称 | BAY-1797 |
包装规格 | 1MG |
CAS编号 | 2055602-83-8 |
别名 | BAY-1797 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by HPLC ,;NMR (Conforms)
分子式:C20H17ClN2O4S
分子量:416.88
溶剂:DMSO (>25 mg/ml)
性状:Pale brown solid
存储:-20°C
Activity (short version):P2X4 antagonist
Function / Pharmacology:BAY-1797 (2055602-83-8) is a selective P2X4 receptor antagonist (IC50 = 211 nM HEK cellular assay; P2X4 calcium influx based assays – hIC50 = 108 nM, mIC50 = 112 nM, rIC50 = 233 nM).1 Displayed antinociceptive and anti-inflammatory effects in mouse CFA inflammatory pain models.?
分子式:C20H17ClN2O4S
分子量:416.88
溶剂:DMSO (>25 mg/ml)
性状:Pale brown solid
存储:-20°C
Activity (short version):P2X4 antagonist
Function / Pharmacology:BAY-1797 (2055602-83-8) is a selective P2X4 receptor antagonist (IC50 = 211 nM HEK cellular assay; P2X4 calcium influx based assays – hIC50 = 108 nM, mIC50 = 112 nM, rIC50 = 233 nM).1 Displayed antinociceptive and anti-inflammatory effects in mouse CFA inflammatory pain models.?