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(R)-PFI-2 HCl
- 英文名称:(R)-PFI-2 HCl
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11078
- cas:1627607-87-7
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11078 |
用途 | 科研检测 |
英文名称 | (R)-PFI-2 HCl |
包装规格 | 1MG |
CAS编号 | 1627607-87-7 |
别名 | (R)-PFI-2 HCl |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC;NMR (Conforms)
分子式:C23H25F4N3O3S HCl
分子量:535.98
溶剂:DMSO (>25 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):Methyltransferase SETD7 inhibitor
Function / Pharmacology:Potent (IC50 = 2nM) and selective SAM-dependent inhibitor of the lysine methyltransferase SETD7.1 It alters Hippo pathway signaling in MCF7 cells by altering YAP nuclear localization in a SETD7-dependent manner.
分子式:C23H25F4N3O3S HCl
分子量:535.98
溶剂:DMSO (>25 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):Methyltransferase SETD7 inhibitor
Function / Pharmacology:Potent (IC50 = 2nM) and selective SAM-dependent inhibitor of the lysine methyltransferase SETD7.1 It alters Hippo pathway signaling in MCF7 cells by altering YAP nuclear localization in a SETD7-dependent manner.