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CPI203
- 英文名称：CPI203
- 品牌：WYTSCI
- 产地：进口
- 型号：1MG
- 货号：WT-AY-B11089
- cas：1446144-04-2
- 价格： ￥1/mg
- 发布日期： 2025-04-10
- 更新日期： 2025-07-15
产品详请
| 产地 | 进口 |
| 品牌 | WYTSCI |
| 货号 | WT-AY-B11089 |
| 用途 | 科研检测 |
| 英文名称 | CPI203 |
| 包装规格 | 1MG |
| CAS编号 | 1446144-04-2 |
| 别名 | CPI203 |
| 纯度 | 98+% |
| 分子式 | |
| 是否进口 | 是 |
纯度:98% by HPLC;NMR (Conforms)
分子式:C19H18ClN5OS
分子量:399.9
溶剂:DMSO (>25 mg/ml)
性状:White to off-white solid
存储:-20°C
Activity (short version):BET bromodomain inhibitor
Function / Pharmacology:CPI203, a JQ1 analog, is a potent and selective inhibitor of the BET bromodomain BRD4 (IC50 = 26 nM).1 It helps promote the maintenance of hematopoietic stem cells via repression of Myc expression.2 CPI203 reversibly suppressed intestinal stem cell differentiation in a mouse model.3 It enhanced the expansion of human cord blood hematopoietic stem cells without losing cell viability.4 CPI203 displays synergistic antitumor activity with various agents including lenalidomide5, bortezomib6, and PARP inhibitors7.
分子式:C19H18ClN5OS
分子量:399.9
溶剂:DMSO (>25 mg/ml)
性状:White to off-white solid
存储:-20°C
Activity (short version):BET bromodomain inhibitor
Function / Pharmacology:CPI203, a JQ1 analog, is a potent and selective inhibitor of the BET bromodomain BRD4 (IC50 = 26 nM).1 It helps promote the maintenance of hematopoietic stem cells via repression of Myc expression.2 CPI203 reversibly suppressed intestinal stem cell differentiation in a mouse model.3 It enhanced the expansion of human cord blood hematopoietic stem cells without losing cell viability.4 CPI203 displays synergistic antitumor activity with various agents including lenalidomide5, bortezomib6, and PARP inhibitors7.
