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Ki8751
- 英文名称：Ki8751
- 品牌：WYTSCI
- 产地：进口
- 型号：1MG
- 货号：WT-AY-B11194
- cas：228559-41-9
- 价格： ￥1/mg
- 发布日期： 2025-04-10
- 更新日期： 2025-05-23
产品详请
| 产地 | 进口 |
| 品牌 | WYTSCI |
| 货号 | WT-AY-B11194 |
| 用途 | 科研检测 |
| 英文名称 | Ki8751 |
| 包装规格 | 1MG |
| CAS编号 | 228559-41-9 |
| 别名 | Ki8751 |
| 纯度 | 98+% |
| 分子式 | |
| 是否进口 | 是 |
纯度:>98% by HPLC;NMR (Conforms)
分子式:C24H18F3N3O4
分子量:469.42
溶剂:DMSO (15 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):VEGFR2 inhibitor
Function / Pharmacology:Very potent (IC50 = 0.9 nM) inhibitor of vascular endothelial growth factor receptor 2 (VEGFR-2).1 It also inhibited PDGFRα (IC50 = 67 nM), c-Kit (IC50 = 40 nM), and FGFR2 (IC50 = 170 nM). Ki8751 completely suppressed HUVEC growth at 1 nM. Ki8751 completely inhibited tumor growth in LC-6 human tumor xenografts @ 5mg/kg. Ki8751 displayed anti-influenza A and B activity via disruption of virus entry in a PDGFR?/GM3-dependent manner.2
分子式:C24H18F3N3O4
分子量:469.42
溶剂:DMSO (15 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):VEGFR2 inhibitor
Function / Pharmacology:Very potent (IC50 = 0.9 nM) inhibitor of vascular endothelial growth factor receptor 2 (VEGFR-2).1 It also inhibited PDGFRα (IC50 = 67 nM), c-Kit (IC50 = 40 nM), and FGFR2 (IC50 = 170 nM). Ki8751 completely suppressed HUVEC growth at 1 nM. Ki8751 completely inhibited tumor growth in LC-6 human tumor xenografts @ 5mg/kg. Ki8751 displayed anti-influenza A and B activity via disruption of virus entry in a PDGFR?/GM3-dependent manner.2
