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CPTH2
- 英文名称:CPTH2
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11259
- cas:357649-93-5
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-07-11
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11259 |
用途 | 科研检测 |
英文名称 | CPTH2 |
包装规格 | 1MG |
CAS编号 | 357649-93-5 |
别名 | CPTH2 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by TLC [10% ethyl acetate in hexanes / Rf: 0.32];NMR (Conforms)
分子式:C14H14ClN3S
分子量:291.80
溶剂:DMSO (25 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):HAT inhibitor
Function / Pharmacology:CPTH2 is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.8 mM). In vitro, the HAT inhibitory activity of CPTH2 was caused via bridge-interaction with histone H3. It’s in vivo activity may involve more histonic and/or non-histonic Gcn5p substrates.
分子式:C14H14ClN3S
分子量:291.80
溶剂:DMSO (25 mg/ml)
性状:White solid
存储:-20°C
Activity (short version):HAT inhibitor
Function / Pharmacology:CPTH2 is a selective inhibitor of the histone acetyltransferase Gcn5P both in vitro and in vivo (IC50 = 0.8 mM). In vitro, the HAT inhibitory activity of CPTH2 was caused via bridge-interaction with histone H3. It’s in vivo activity may involve more histonic and/or non-histonic Gcn5p substrates.