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ML418
- 英文名称:ML418
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11339
- cas:1928763-08-9
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-05-23
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11339 |
用途 | 科研检测 |
英文名称 | ML418 |
包装规格 | 1MG |
CAS编号 | 1928763-08-9 |
别名 | ML418 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:>98% by HPLC;NMR (Conforms)
分子式:C19H24ClN3O3
分子量:377.87
溶剂:DMSO (8 mg/ml, with warming)
性状:White solid
存储:-20°C
Activity (short version):Kir7.1/6.2 blocker
Function / Pharmacology:ML418 is a blocker of the inward rectifier potassium channels Kir7.1 (IC50 = 310nM) and Kir6.2 (equipotent) with metabolic and pharmacokinetic parameters suitable for in vivo research.1 Greater than 23-fold selectivity over Kir1.1, Kir2.1, Kir2.2, Kir2.3, Kir4.1.
分子式:C19H24ClN3O3
分子量:377.87
溶剂:DMSO (8 mg/ml, with warming)
性状:White solid
存储:-20°C
Activity (short version):Kir7.1/6.2 blocker
Function / Pharmacology:ML418 is a blocker of the inward rectifier potassium channels Kir7.1 (IC50 = 310nM) and Kir6.2 (equipotent) with metabolic and pharmacokinetic parameters suitable for in vivo research.1 Greater than 23-fold selectivity over Kir1.1, Kir2.1, Kir2.2, Kir2.3, Kir4.1.