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AZD1152-HQPA
- 英文名称:AZD1152-HQPA
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11414
- cas:722544-51-6
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-04-30
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11414 |
用途 | 科研检测 |
英文名称 | AZD1152-HQPA |
包装规格 | 1MG |
CAS编号 | 722544-51-6 |
别名 | AZD1152-HQPA |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by HPLC;NMR (Conforms)
分子式:C26H30FN7O3
分子量:507.56
溶剂:DMSO (15 mg/ml)
性状:Yellow solid
存储:-20°C
Activity (short version):Aurora B kinase inhibitor
Function / Pharmacology:AZD1152-HQPA is a potent and highly selective inhibitor of Aurora B.1 Aurora B Ki = 0.36 nM; Aurora A Ki = 1,369 nM.2 It inhibits the growth of tumors in multiple cancer models.3-6 Excessive ROS generation7 and upregulated tumor suppressor miRNAs8 have been proposed as a novel mechanisms of cytotoxicity of AZD1152-HQPA.
分子式:C26H30FN7O3
分子量:507.56
溶剂:DMSO (15 mg/ml)
性状:Yellow solid
存储:-20°C
Activity (short version):Aurora B kinase inhibitor
Function / Pharmacology:AZD1152-HQPA is a potent and highly selective inhibitor of Aurora B.1 Aurora B Ki = 0.36 nM; Aurora A Ki = 1,369 nM.2 It inhibits the growth of tumors in multiple cancer models.3-6 Excessive ROS generation7 and upregulated tumor suppressor miRNAs8 have been proposed as a novel mechanisms of cytotoxicity of AZD1152-HQPA.