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T-10418
- 英文名称:T-10418
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11458
- cas:1608784-68-4
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-04-30
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11458 |
用途 | 科研检测 |
英文名称 | T-10418 |
包装规格 | 1MG |
CAS编号 | 1608784-68-4 |
别名 | T-10418 |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by HPLC;NMR (Conforms)
分子式:C22H20N2O4
分子量:376.14
溶剂:DMSO (>65 mg/ml)
性状:Off-white solid
存储:-20°C
Activity (short version):G2A agonist
Function / Pharmacology:T-10418 is a potent (EC50 = 820 nM) and selective (against 300 non-olfactory GPCRs) agonist of G2 accumulation protein (G2A; GPR132). At 100 nM, T-10418 resulted in 244% TRPV1 sensitization in mouse sensory neurons. T-10418 is an interesting new chemical tool to study G2A biology.
分子式:C22H20N2O4
分子量:376.14
溶剂:DMSO (>65 mg/ml)
性状:Off-white solid
存储:-20°C
Activity (short version):G2A agonist
Function / Pharmacology:T-10418 is a potent (EC50 = 820 nM) and selective (against 300 non-olfactory GPCRs) agonist of G2 accumulation protein (G2A; GPR132). At 100 nM, T-10418 resulted in 244% TRPV1 sensitization in mouse sensory neurons. T-10418 is an interesting new chemical tool to study G2A biology.