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PD 123319 ditrifluoroacetate
- 英文名称:PD 123319 ditrifluoroacetate
- 品牌:WYTSCI
- 产地:进口
- 型号:1MG
- 货号:WT-AY-B11476
- cas:136676-91-0
- 价格: ¥1/mg
- 发布日期: 2025-04-10
- 更新日期: 2025-04-30
产品详请
产地 | 进口 |
品牌 | WYTSCI |
货号 | WT-AY-B11476 |
用途 | 科研检测 |
英文名称 | PD 123319 ditrifluoroacetate |
包装规格 | 1MG |
CAS编号 | 136676-91-0 |
别名 | PD 123319 ditrifluoroacetate |
纯度 | 98+% |
分子式 | |
是否进口 | 是 |
纯度:98% by HPLC;NMR (Conforms)
分子式:C31H32N4O3·2CF3CO2H
分子量:736.66
溶剂:DMSO (>25 mg/ml) Water (>25 mg/ml)
性状:Yellow solid
存储:-20°C
Activity (short version):Angiotensin II type II antagonist
Function / Pharmacology:Potent (IC50 = 34 nM) and selective non-peptide angiotensin II type 2 (AT2) antagonist.1 Ameliorated symptoms of 2,4-dinitrobenzenesulfonic-induced colitis in rats via inhibition of NF-kB activation.2 PD123319 displayed protective effects in ischemia-reperfusion injury and oxidative damage in rat hearts.3
分子式:C31H32N4O3·2CF3CO2H
分子量:736.66
溶剂:DMSO (>25 mg/ml) Water (>25 mg/ml)
性状:Yellow solid
存储:-20°C
Activity (short version):Angiotensin II type II antagonist
Function / Pharmacology:Potent (IC50 = 34 nM) and selective non-peptide angiotensin II type 2 (AT2) antagonist.1 Ameliorated symptoms of 2,4-dinitrobenzenesulfonic-induced colitis in rats via inhibition of NF-kB activation.2 PD123319 displayed protective effects in ischemia-reperfusion injury and oxidative damage in rat hearts.3